Harald H?bner : rechercher sur Z-Library

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1

Discovery of Highly Potent and Neurotensin Receptor 2 Selective Neurotensin Mimetics

Einsiedel, Jürgen, Held, Cornelia, Hervet, Maud, Plomer, Manuel, Tschammer, Nuska, Hübner, Harald, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 1.00 MB

english, 2011

2

Azepino- and Diazepinoindoles: Synthesis and Dopamine Receptor Binding Profiles

Johannes Kraxner, Harald H?bner, Peter Gmeiner

Journal:

Archiv der Pharmazie

Année:

2000

Langue:

english

Fichier:

PDF, 97 KB

english, 2000

3

Highly Potent 5-Aminotetrahydropyrazolopyridines: Enantioselective Dopamine D3 Receptor Binding, Functional Selectivity, and Analysis of Receptor−Ligand Interactions

Tschammer, Nuska, Elsner, Jan, Goetz, Angela, Ehrlich, Katharina, Schuster, Stefan, Ruberg, Miriam, Kühhorn, Julia, Thompson, Dawn, Whistler, Jennifer, Hübner, Harald

Journal:

Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 1.14 MB

english, 2011

4

Bivalent Dopamine D 2 Receptor Ligands: Synthesis and Binding Properties

Kühhorn, Julia, Hübner, Harald, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2011

Langue:

english

Fichier:

PDF, 1.02 MB

english, 2011

5

Novel Pyridylmethylamines as Highly Selective 5-HT 1A Superagonists

Bollinger, Stefan, Hübner, Harald, Heinemann, Frank W., Meyer, Karsten, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 1.08 MB

english, 2010

6

Dopamine D 2 , D 3 , and D 4 Selective Phenylpiperazines as Molecular Probes To Explore the Origins of Subtype Specific Receptor Binding

Ehrlich, Katharina, Götz, Angela, Bollinger, Stefan, Tschammer, Nuska, Bettinetti, Laura, Härterich, Steffen, Hübner, Harald, Lanig, Harald, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 3.72 MB

english, 2009

7

Engineering a GPCR−Ligand Pair That Simulates the Activation of D 2L by Dopamine

Tschammer, Nuska, Dörfler, Miriam, Hübner, Harald, Gmeiner, Peter

Journal:

ACS Chemical Neuroscience

Année:

2010

Langue:

english

Fichier:

PDF, 1.68 MB

english, 2010

8

1,1′-Disubstituted Ferrocenes as Molecular Hinges in Mono- and Bivalent Dopamine Receptor Ligands

Huber, Daniela, Hübner, Harald, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2009

Langue:

english

Fichier:

PDF, 1.04 MB

english, 2009

9

Novel D3 Selective Dopaminergics Incorporating Enyne Units as Nonaromatic Catechol Bioisosteres: Synthesis, Bioactivity, and Mutagenesis Studies

Dörfler, Miriam, Tschammer, Nuska, Hamperl, Katharina, Hübner, Harald, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2008

Langue:

english

Fichier:

PDF, 341 KB

english, 2008

10

Synthesis of a 68 Ga-Labeled Peptoid−Peptide Hybrid for Imaging of Neurotensin Receptor Expression in Vivo

Maschauer, Simone, Einsiedel, Jürgen, Hocke, Carsten, Hübner, Harald, Kuwert, Torsten, Gmeiner, Peter, Prante, Olaf

Journal:

ACS Medicinal Chemistry Letters

Année:

2010

Langue:

english

Fichier:

PDF, 1.65 MB

english, 2010

11

Bioisosteric Replacement Leading to Biologically Active [2.2]Paracyclophanes with Altered Binding Profiles for Aminergic G-Protein-Coupled Receptors

Skultety, Marika, Hübner, Harald, Löber, Stefan, Gmeiner, Peter

Journal:

Journal of Medicinal Chemistry

Année:

2010

Langue:

english

Fichier:

PDF, 1.09 MB

english, 2010

12

Selective and Wash-Resistant Fluorescent Dihydrocodeinone Derivatives Allow Single-Molecule Imaging of Î¼-Opioid Receptor Dimerization

Gentzsch, Christian, Seier, Kerstin, Drakopoulos, Antonios, Jobin, Marie-Lise, LanoiselÃ©e, Yann, Koszegi, Zsombor, Maurel, Damien, Sounier, RÃ©my, HÃ¼bner, Harald, Gmeiner, Peter, Granier, SÃ©bastien

Journal:

Angewandte Chemie International Edition

Année:

2020

Langue:

english

Fichier:

PDF, 1.61 MB

english, 2020

13

Investigation of inactive state Îº opioid receptor homodimerization via single molecule microscopy using new antagonistic fluorescent probes

Drakopoulos, Antonios, Koszegi, Zsombor, LanoiselÃ©e, Yann, HÃ¼bner, Harald, Gmeiner, Peter, Calebiro, Davide, Decker, Michael

Journal:

Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 1.66 MB

2020

14

Selective and WashâResistant Fluorescent Dihydrocodeinone Derivatives Allow SingleâMolecule Imaging of Î¼âOpioid Receptor Dimerization

Gentzsch, Christian, Seier, Kerstin, Drakopoulos, Antonios, Jobin, MarieâLise, LanoiselÃ©e, Yann, Koszegi, Zsombor, Maurel, Damien, Sounier, RÃ©my, HÃ¼bner, Harald, Gmeiner, Peter, Granier, SÃ©basti

Journal:

Angewandte Chemie

Année:

2020

Langue:

german

Fichier:

PDF, 1.56 MB

german, 2020

15

Regiospecific introduction of halogens on the 2-aminobiphenyl subunit leads to highly potent and selective M3 muscarinic acetylcholine receptor antagonists and weak inverse agonists

Fischer, Oliver, Hofmann, Josefa, Rampp, Hannelore, Kaindl, Jonas, Pratsch, Gerald, Bartuschat, Amelie, Taudte, Regina Verena, Fromm, Martin Friedrich, HÃ¼bner, Harald, Gmeiner, Peter, Heinrich, Marku

Journal:

Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 977 KB

english, 2020

16

Red-emitting dibenzodiazepinone derivatives as fluorescent dualsteric probes for the muscarinic acetylcholine M 2 receptor

She, Xueke, Pegoli, Andrea, Gruber, Corinna G., Wifling, David, Carpenter, Jessica, HÃ¼bner, Harald, Chen, Mengya, Wan, Jianfei, Bernhardt, GÃ¼nther, Gmeiner, Peter, Holliday, Nicholas D., Keller, Max

Journal:

Journal of Medicinal Chemistry

Année:

2020

Langue:

english

Fichier:

PDF, 5.98 MB

english, 2020

17

Synthesis, biological evaluation and radiosynthesis of buprenorphineâderived phenylazocarboxamides as novel Î¼âopioid receptor ligands

KrÃ¼ll, Jasmin, Fehler, Stefanie K., Hofmann, Laura, Nebel, Natascha, Maschauer, Simone, Prante, Olaf, Gmeiner, Peter, Lanig, Harald, HÃ¼bner, Harald, Heinrich, Markus Rolf

Journal:

Année:

2020

Fichier:

PDF, 1.91 MB

2020

18

T215. THE ANTIPSYCHOTIC ACTION OF HALOPERIDOL IN PSYCHOTIC-LIKE RATS REQUIRES PRESYNAPTIC VESICULAR ACCUMULATION

MÃ¼ller, Christian, Weiss, Eva-Maria, Hellmann, Jan, Dahlmanns, Jana, Kalinichenko, Liubov, Alzheimer, Christian, LÃ¶ber, Stefan, HÃ¼bner, Harald, Kornhuber, Johannes, Gmeiner, Peter, GrÃ¶mer, Teja, U

Journal:

Schizophrenia Bulletin

Année:

2020

Fichier:

PDF, 80 KB

2020

19

Discovery of Novel Nonpeptidic PAR2 Ligands

KlÃ¶sel, Ilona, Schmidt, Maximilian F., Kaindl, Jonas, HÃ¼bner, Harald, Weikert, Dorothee, Gmeiner, Peter

Journal:

ACS Medicinal Chemistry Letters

Année:

2020

Fichier:

PDF, 596 KB

2020

20

An allosteric modulator binds to a conformational hub in the Î²2 adrenergic receptor

Liu, Xiangyu, Kaindl, Jonas, Korczynska, Magdalena, StÃ¶Ãel, Anne, Dengler, Daniela, Stanek, Markus, HÃ¼bner, Harald, Clark, Mary J., Mahoney, Jake, Matt, Rachel Ann, Xu, Xinyu, Hirata, Kunio, Shoich

Journal:

Nature Chemical Biology

Année:

2020

Fichier:

PDF, 2.65 MB

2020

21

Structure-based development of a subtype-selective orexin 1 receptor antagonist

Hellmann, Jan, Drabek, MatthÃ¤us, Yin, Jie, Gunera, Jakub, PrÃ¶ll, Theresa, Kraus, Frank, Langmead, Christopher J., HÃ¼bner, Harald, Weikert, Dorothee, Kolb, Peter, Rosenbaum, Daniel M., Gmeiner, Pete

Journal:

Proceedings of the National Academy of Sciences

Année:

2020

Fichier:

PDF, 2.20 MB

2020

22

Radiosynthesis and evaluation of 18F-labeled dopamine D4-receptor ligands

Willmann, Michael, Ermert, Johannes, Prante, Olaf, HÃ¼bner, Harald, Gmeiner, Peter, Neumaier, Bernd

Journal:

Nuclear Medicine and Biology

Année:

2020

Fichier:

PDF, 3.87 MB

2020

23

Pharmacological characterization of low-to-moderate affinity opioid receptor agonists and brain imaging with 18F-labeled derivatives in rats.

Ott, Julian J, Spilhaug, Mona M., Maschauer, Simone, Rafique, Waqas, Jakobsson, Jimmy E., Hartvig, Karoline, HÃ¼bner, Harald, Gmeiner, Peter, Prante, Olaf, Riss, Patrick J

Journal:

Journal of Medicinal Chemistry

Année:

2020

Fichier:

PDF, 5.19 MB

2020

24

Binding pathway determines norepinephrine selectivity for the human Î²1AR over Î²2AR

Xu, Xinyu, Kaindl, Jonas, Clark, Mary J., HÃ¼bner, Harald, Hirata, Kunio, Sunahara, Roger K., Gmeiner, Peter, Kobilka, Brian K., Liu, Xiangyu

Journal:

Année:

2020

Fichier:

PDF, 3.34 MB

2020